I-protein inhibitor iyizinhlayiyana ezijoyina i-catalyst, ivimbela isenzo sayo. Ama-Catalysts, okungamaprotheni asiza impendulo eyinhlanganisela eyisisekelo phakade, asebenza ngokushintsha izinhlayiya ze-substrate zibe imikhiqizo.[1] Ikhemikhali ifeza lokhu ngokukhawulela i-substrate endaweni yayo eguquguqukayo, indawo ethile esheshisa isinyathelo esinzima kakhulu sokuphendula.


I-protein inhibitor ilamula kulo mjikelezo ngomunye noma omunye ngokukhawula endaweni eguquguqukayo yekhemikhali, igcina i-substrate ingakhawuleli, noma ibeke imingcele endaweni eyodwa ngaphezulu kwenhlanganisela, idikibalise i-catalyst ye-catalyst yempendulo. Ama-inhibitors angabonisa imikhawulo ehlehliswayo noma engenakuhlehliswa. Ama-Irreversible inhibitors enza isibopho esihlanganisiwe neprotheni, ayicindezele kuze kube yilapho isibopho siphulwa. 


Okunye, ama-reversible inhibitors abopha ngokungabambeki futhi angakwazi ukuzihlukanisa ngokushesha ne-catalyst, avumele iphrotheni ukuthi iqhubeke namandla ayo. Kuya ngokuthi ajoyina ikhemikhali, i-compound substrate complex, noma kokubili, ama-reversible inhibitors adala izinhlobo ezahlukene zokuzithiba.


Ama-inhibitors

  • I-Glecaprevir

    CAS: 1365970-03-1
    Ukubukeka: Impushana emhlophe ukuya kokumhlophe
    I-Assay: 98%
    Igama Brand: YIHUI
    Ukupakisha: 1g;10g;100g
    Ikhono Lokuhlinzeka: 2000g ngenyangaImpilo yeshelufu: Iminyaka emibili
    Isicelo: ucwaningo lwelebhu
    Inkokhelo: T/T, LC noma DA
    Isampula: iyatholakala
    Isikhathi Sokulethwa: Isitokwe Esilungile Esitolo Sendawo, izinsuku ezingu-1-3
    Ngokushesha futhi Kuvikelekile Ukuthunyelwa
    Umsuka: China
    Ukuthumela: DHL,FedEx,TNT,EMS,Ngolwandle,Ngomoya
    Izitifiketi: ISO9001, ISO22000, HACCP, HALAL, KOSHER
    Ayikwazi ukudayisela abantu ngabanye

  • I-Finerenone API

    I-CAS Cha: 1050477-31-0
    Ukubukeka: Impushana ecwebezelayo emhlophe ukuya kokuphuzi
    Okujwayelekile: endlini
    Ikhono Lokuhlinzeka: 5000g ngenyanga
    Ubumsulwa: ≥99%
    Inkokhelo: T/T, LC noma DA
    Isikhathi Sokulethwa: Isitokwe Esilungile Esitolo Sendawo, izinsuku ezingu-1-3
    Umsuka: China
    Ukuthumela: DHL, FedEx, TNT, EMS, By Sea, By Air
    Ayikwazi ukudayisela abantu ngabanye

  • I-Pyrilutamide

    I-CAS Cha: 1272719-00-2
    Ukubukeka: impushana emhlophe ukuya kokuphuzi ngokukhanyayo
    Okujwayelekile: endlini
    Ikhono Lokuhlinzeka: 1000g ngenyanga
    Ubumsulwa: ≥99%
    Inkokhelo: T/T, LC noma DA
    Isikhathi Sokulethwa: Isitokwe Esilungile Esitolo Sendawo, izinsuku ezingu-1-3
    Umsuka: China
    Ukuthumela: DHL, FedEx, TNT, EMS, By Sea, By Air
    Ayikwazi ukudayisela abantu ngabanye

  • I-Setipiprant powder

    I-CAS Cha: 866460-33-5
    Ukubukeka: impushana ephuzi ekhanyayo
    Okujwayelekile: endlini
    Ikhono Lokuhlinzeka: 1000g ngenyanga
    Ubumsulwa: ≥99%
    Inkokhelo: T/T, LC noma DA
    Isikhathi Sokulethwa: Isitokwe Esilungile Esitolo Sendawo, izinsuku ezingu-1-3
    Umsuka: China
    Ukuthumela: DHL, FedEx, TNT, EMS, By Sea, By Air
    Ayikwazi ukudayisela abantu ngabanye

  • I-clascoterone powder

    I-CAS Cha: 19608-29-8
    Ukubukeka: impushana emhlophe ukuya kokuphuzi ngokukhanyayo
    Okujwayelekile: endlini
    Supply Amandla: 100kg ngenyanga
    Ubumsulwa: ≥99%
    Inkokhelo: T/T, LC noma DA
    Isikhathi Sokulethwa: Isitokwe Esilungile Esitolo Sendawo, izinsuku ezingu-1-3
    Umsuka: China
    Ukuthumela: DHL, FedEx, TNT, EMS, By Sea, By Air
    Ayikwazi ukudayisela abantu ngabanye

  • I-AZD 8055

    I-CAS Cha: 1009298-09-2
    Ukubukeka: Okuqinile okuphuzi kuya kokuphuzi
    Okujwayelekile: endlini
    Ikhono Lokuhlinzeka: 1000g ngenyanga
    Ubumsulwa: ≥99%
    Inkokhelo: T/T, LC noma DA
    Isikhathi Sokulethwa: Isitokwe Esilungile Esitolo Sendawo, izinsuku ezingu-1-3
    Umsuka: China
    Ukuthumela: DHL, FedEx, TNT, EMS, By Sea, By Air
    Ayikwazi ukudayisela abantu ngabanye

  • I-AZD 1480

    I-CAS Cha: 935666-88-9
    Ukubukeka: okumhlophe kuya ku-beige powder
    Okujwayelekile: endlini
    Ikhono Lokuhlinzeka: 1000g ngenyanga
    Ubumsulwa: ≥99%
    Inkokhelo: T/T, LC noma DA
    Isikhathi Sokulethwa: Isitokwe Esilungile Esitolo Sendawo, izinsuku ezingu-1-3
    Umsuka: China
    Ukuthumela: DHL, FedEx, TNT, EMS, By Sea, By Air
    Ayikwazi ukudayisela abantu ngabanye

  • I-Alagebrium Chloride

    I-CAS Cha: 341028-37-3
    Ukubukeka: cishe impushana enombala omhlophe noma omhlophe
    Okujwayelekile: endlini
    Ikhono Lokuhlinzeka: 1000g ngenyanga
    Ubumsulwa: ≥99%
    Inkokhelo: T/T, LC noma DA
    Isikhathi Sokulethwa: Isitokwe Esilungile Esitolo Sendawo, izinsuku ezingu-1-3
    Umsuka: China
    Ukuthumela: DHL, FedEx, TNT, EMS, By Sea, By Air
    Ayikwazi ukudayisela abantu ngabanye

  • EPZ-6438

    I-CAS Cha: 1403254-99-8
    Ukubukeka: I-crystalline powder emhlophe noma emhlophe
    Okujwayelekile: endlini
    Isicelo: Ucwaningo lwelebhu  
    Ikhono Lokuhlinzeka: 1000g ngenyanga
    Ubumsulwa: ≥98%
    Inkokhelo: T/T, LC noma DA
    Isikhathi Sokulethwa: Isitokwe Esilungile Esitolo Sendawo, izinsuku ezingu-1-3
    Umsuka: China
    Ukuthumela: DHL, FedEx, TNT, EMS, By Sea, By Air
    Ayikwazi ukudayisela abantu ngabanye

  • I-Verteporfin API

    I-CAS Cha: 129497-78-5
    Ukubukeka: Okuluhlaza okumnyama kuya kokuqinile okumnyama
    Okujwayelekile: endlini
    Isicelo: Ucwaningo lwelebhu 
    Ikhono Lokuhlinzeka: 100g ngenyanga
    Ubumsulwa: ≥96%
    Inkokhelo: T/T, LC noma DA
    Isikhathi Sokulethwa: Isitokwe Esilungile Esitolo Sendawo, izinsuku ezingu-1-3
    Umsuka: China
    Ukuthumela: DHL, FedEx, TNT, EMS, By Sea, By Air
    Ayikwazi ukudayisela abantu ngabanye

  • I-Vismodegib

    I-CAS Cha: 879085-55-9
    Ukubukeka: Impushana emhlophe noma Ephuzi noma Ikristalu
    Okujwayelekile: endlini
    Isicelo: Anti tumor; anti-umdlavuza 
    Supply Amandla:50kg ngenyanga
    Ubumsulwa: ≥99%
    Inkokhelo: T/T, LC noma DA
    Isikhathi Sokulethwa: Isitokwe Esilungile Esitolo Sendawo, izinsuku ezingu-1-3
    Umsuka: China
    Ukuthumela: DHL, FedEx, TNT, EMS, By Sea, By Air
    Ayikwazi ukudayisela abantu ngabanye

  • I-PLX5622

    Inombolo ye-CAS: 1303420-67-8
    Ukubukeka: Impushana ephuzi ngokuphaphathekile
    Okujwayelekile: I-Enterprise Standard
    Supply Amandla:5000g ngenyanga
    Impilo Yeshelufu: Iminyaka emibili
    Inkokhelo: T/T, LC noma DA
    Isikhathi Sokulethwa: Isitokwe Esilungile Esitolo Sendawo, izinsuku ezingu-1-3
    Umsuka: China
    Ukuthumela: DHL, FedEx, TNT, EMS, By Sea, By Air
    Nikeza abasebenzi baselabhorethri ngezinjongo zocwaningo, hhayi ukudayiselwa iziguli

Amakhasi angu-3 esewonke